ID	activity	Label
acrivastine	88	Substrate-to-Pgp
alprenolol	93	Not-substrate-to-Pgp
amantadine	95	Not-substrate-to-Pgp
amitriptylline	95	Not-substrate-to-Pgp
amprenavir	70	Substrate-to-Pgp
antipyrine	97	Not-substrate-to-Pgp
astemizole	90	Substrate-to-Pgp
atenolol	50	Not-substrate-to-Pgp
biperidine-biperiden	100	Not-substrate-to-Pgp
bromocriptine	30	Not-substrate-to-Pgp
bufuralol	na	Not-substrate-to-Pgp
buspirone	87	Not-substrate-to-Pgp
carbamazepine	70	Not-substrate-to-Pgp
cetirizine	60	Substrate-to-Pgp
chloroquine	100	Substrate-to-Pgp
chlorpheniramine	34	Not-substrate-to-Pgp
chlorpromazine	96	Substrate-to-Pgp
chlorprothixene	na	Not-substrate-to-Pgp
cimetidine	64	Substrate-to-Pgp
clarithromycin	100	Substrate-to-Pgp
clemastine funurate	90	Not-substrate-to-Pgp
clomipramine	80	Not-substrate-to-Pgp
clonidine	100	Not-substrate-to-Pgp
colchicine	44	Substrate-to-Pgp
cyclobenzaprine	100	Not-substrate-to-Pgp
cyclosporin	40	Substrate-to-Pgp
daunorubicin	10	Substrate-to-Pgp
desipramine	100	Not-substrate-to-Pgp
dexamethasone	81	Substrate-to-Pgp
diltiazem	90	Substrate-to-Pgp
diphenhydramine	50	Not-substrate-to-Pgp
dipyridamole	60	Substrate-to-Pgp
domperidone	93	Substrate-to-Pgp
doxapram	60	Not-substrate-to-Pgp
doxepin	27	Not-substrate-to-Pgp
doxorubicin	12	Not-substrate-to-Pgp
doxylamine	na	Not-substrate-to-Pgp
eletriptan	50	Substrate-to-Pgp
emetine	na	Substrate-to-Pgp
erythromycin	35	Substrate-to-Pgp
etoposide	50	Substrate-to-Pgp
famciclovir	60	Substrate-to-Pgp
flumazenil	95	Not-substrate-to-Pgp
fluoxetine	95	Not-substrate-to-Pgp
flurazepam	100	Not-substrate-to-Pgp
fluvoxamine	53	Not-substrate-to-Pgp
guanbenz	79	Not-substrate-to-Pgp
guanfacine	80	Not-substrate-to-Pgp
haloperidol	100	Not-substrate-to-Pgp
hoechst 33342	na	Substrate-to-Pgp
imipramine	100	Not-substrate-to-Pgp
indinavir	62.5	Substrate-to-Pgp
indomethacine	100	Not-substrate-to-Pgp
itraconazole	85	Not-substrate-to-Pgp
ketamine	na	Not-substrate-to-Pgp
ketoconazole	76	Substrate-to-Pgp
labetalol	14	Substrate-to-Pgp
levomepromazine-methotrimeprazine	21	Substrate-to-Pgp
lidocaine	35	Not-substrate-to-Pgp
loperamide	40	Substrate-to-Pgp
loratadine	90	Substrate-to-Pgp
lorcainide	na	Not-substrate-to-Pgp
mannitol	15	Not-substrate-to-Pgp
maprotiline	95	Not-substrate-to-Pgp
mebendazole	5	Substrate-to-Pgp
mephentermine	na	Not-substrate-to-Pgp
meprobamate	90	Not-substrate-to-Pgp
mequitazine	na	Substrate-to-Pgp
metergoline	na	Not-substrate-to-Pgp
methotrexate	65	Not-substrate-to-Pgp
methotrimeprazine(levomeprazine)	21	Substrate-to-Pgp
methysergide	13	Substrate-to-Pgp
metoprolol	98	Not-substrate-to-Pgp
mexilitene	100	Not-substrate-to-Pgp
midazolam	36	Substrate-to-Pgp
mitoxantrone	85	Substrate-to-Pgp
monensin	na	Substrate-to-Pgp
nalbuphine	12	Substrate-to-Pgp
naloxone	95	Not-substrate-to-Pgp
naltrexone	100	Not-substrate-to-Pgp
nelfinavir	78	Substrate-to-Pgp
neostigmine	10	Substrate-to-Pgp
nicardipine	95	Substrate-to-Pgp
nifedipine	45	Substrate-to-Pgp
nitrazepam	78	Not-substrate-to-Pgp
nitrendipine	15	Not-substrate-to-Pgp
nordazepam	na	Not-substrate-to-Pgp
nortriptyline	100	Not-substrate-to-Pgp
noscapine	100	Not-substrate-to-Pgp
oxprenolol	95	Not-substrate-to-Pgp
paclitaxel	6	Substrate-to-Pgp
perphenazine	70	Not-substrate-to-Pgp
pheniramine	77	Not-substrate-to-Pgp
pirenzepine	25	Substrate-to-Pgp
practolol	100	Not-substrate-to-Pgp
prazosin	57	Substrate-to-Pgp
procyclidine	100	Not-substrate-to-Pgp
progabide	60	Not-substrate-to-Pgp
promazine	40	Not-substrate-to-Pgp
promethazine	25	Not-substrate-to-Pgp
propranolol	90	Not-substrate-to-Pgp
protriptyline	90	Substrate-to-Pgp
puromycin	na	Substrate-to-Pgp
pyridostigmine	10	Not-substrate-to-Pgp
quinidine	80	Substrate-to-Pgp
ranitidine	52	Not-substrate-to-Pgp
reserpine	50	Substrate-to-Pgp
risperidone	70	Substrate-to-Pgp
ritonavir	68	Substrate-to-Pgp
saquinavir	4	Substrate-to-Pgp
scopolamine	95	Not-substrate-to-Pgp
selegiline	100	Not-substrate-to-Pgp
sulfasalazine	59	Not-substrate-to-Pgp
sumatriptan	14	Not-substrate-to-Pgp
tacrine	17	Not-substrate-to-Pgp
terfenadine	70	Substrate-to-Pgp
trazodone	90	Not-substrate-to-Pgp
triamterene	54	Not-substrate-to-Pgp
trimethoprim	97	Substrate-to-Pgp
trimipramine	100	Substrate-to-Pgp
verapamil	28	Substrate-to-Pgp
vinblastine	5	Substrate-to-Pgp
vincristine	na	Substrate-to-Pgp
vinorelbine	27	Substrate-to-Pgp
warfarin	98	Not-substrate-to-Pgp
yohimbine	na	Not-substrate-to-Pgp
zimeldine	na	Not-substrate-to-Pgp
zolmitriptan	91.5	Not-substrate-to-Pgp
zolpidem	100	Substrate-to-Pgp
